Ligand induced changes of the 18kDa translocator protein in a lipid bilayer

DOI

The proposed experiments will investigate conformational changes of the 18kDa translocator protein (TSPO) in a lipid bilayer using neutron reflectometry at the solid-liquid interface. The TSPO will be immobilised to a solid surface and a lipid bilayer formed around the protein layer. Preliminary data indicates that interaction of the protein with its ligand PK11195 induces a conformational change, possibly the formation of a channel. The aim of the proposed experiment is to investigate channel formation by using neutrons to detect increased water content in the protein-lipid bilayer as a result of ligand binding. In addition, there is evidence that TSPO acts as a cholesterol recognition site and transporter. Hence, we will also examine changes associated with cholesterol binding. We hope to contribute to a better understanding of structure-function relationships of the TSPO.

Identifier
DOI https://doi.org/10.5286/ISIS.E.24088332
Metadata Access https://icatisis.esc.rl.ac.uk/oaipmh/request?verb=GetRecord&metadataPrefix=oai_datacite&identifier=oai:icatisis.esc.rl.ac.uk:inv/24088332
Provenance
Creator Professor Richard Banati; Miss Claire Hatty
Publisher ISIS Neutron and Muon Source
Publication Year 2014
Rights CC-BY Attribution 4.0 International; https://creativecommons.org/licenses/by/4.0/
OpenAccess true
Contact isisdata(at)stfc.ac.uk
Representation
Resource Type Dataset
Discipline Photon- and Neutron Geosciences
Temporal Coverage Begin 2011-12-13T05:09:19Z
Temporal Coverage End 2011-12-17T09:29:42Z